TB Research

Research Capstone Experiences: Design, Synthesis, In Silico Analysis, and Assay Development Towards Prokaryotic Proteasome Antagonists

Tony D. Davis, Serena Farnell, Joseph D'Antonio, Juhi Gurtata, Eric Kelly, Mana Halaji Dezfuli, Azim Sama

American Journal of Pharmaceutical Education · 2023-08

Abstract

Herein, we report the development of antagonists of the Mycobacterium tuberculosis prokaryotic proteasome system (PPS) to address drug-resistant tuberculosis infections.

MeSH terms

  • Proteasome
  • In silico
  • Mycobacterium tuberculosis
  • Tuberculosis
  • Computational biology
  • Drug development
  • Biology
  • Microbiology
  • Drug
  • Medicine