TB Research

Quinolone-isoniazid hybrids: synthesis and preliminary <i>in vitro</i> cytotoxicity and anti-tuberculosis evaluation

Richard M. Beteck, Ronnett Seldon, Audrey Jordaan, Digby F. Warner, Heinrich C. Hoppe, Dustin Laming, Lesetja J. Legoabe, Setshaba D. Khanye

MedChemComm · 2019-01

Abstract

A new series of quinolone-isoniazid hybrid compounds were designed, synthesised and studied for their potential anti-mycobacterial tuberculosis activity <italic>in vitro</italic>.

MeSH terms

  • Isoniazid
  • Quinolone
  • Cytotoxicity
  • In vitro
  • Tuberculosis
  • Microbiology
  • Virology
  • Biology
  • Chemistry